Peptide Active Data Details
Basic Peptide Information
DICL ID
DICL_Pep_02458
Ion Channel
Voltage-gated sodium channel type 3 subunit alpha
Peptide Function
Inhibitor
Gene Name
SCN3A
Activity Data (nM)
IC50
2200 nM
Ki
Not available
EC50
Not available
Kd
Not available
Biologically Active
Not specified
Sequence Information
Peptide Sequence
MKVTLIAILTCAALLVLLHTTAAEELEAQEESQLMEVGMPDTELAALDEERIFECSISCEIEKEGNGKKCKPKKCKGGWKCKFNICVKV
Peptide UniProt Accession
Not available
UniParc
Not available
Peptide Synonyms/Alias
μ-TrtX-Ca1a
Peptide Species
C. albostriatus
Peptide Name
Not available
CAS Number
Not available
Experimental Conditions
pH
pH 7.4
Holding Potential (mV)
–110 to -10 mV
Temperature
20–25 °C
Test Method
Patch-clamping
Test Species
Not specified
Binding Information
Binding Site
Not specified
Binding Site Residue
Not specified
Ion Channel Information
Gene Abbreviation (ABB)
VGSCs
Ion Channel UniProt Accession
Source Organism
Rattus norvegicus (Rat)
References & Disease Information
Disease
Not specified
PubChem CID
Not available
URL
Not available
PMID
Patent
Not available